Hyperlipidemia

high cholesterol or triglycerides (fat) levels in blood

Bloodwork  will show elevated lipid levels (cholesterol and triglycerides). If hyperlipidemia is not treated, it can cause arteries to become blocked. If arteries in the heart or brain are blocked it can lead to coronary artery disease or stroke.

When does hyperlipidemia start and how long does it last?

Lorlatinib is most likely to cause hyperlipidemia. On average, hyperlipidemia begins 15 days after starting treatment, and lasts for 15 months.

How serious is hyperlipidemia?

The severity most often experienced is grade 1 or 2 but grade 3 or 4 are possible

How likely is it that I will experience hyperlipidemia?

Lorlatinib: 83% of people require lipid lowering therapy. Alectinib: hyperlipidemia is uncommon. Crizotinib: 5% of people will experience hyperlipidemia.

Prevention Strategies

blood vial with magnifying glass
  • Your healthcare team will monitor blood lipid levels including serum cholesterol and triglyceride.

    Blood lipid levels should be checked:

    • Before starting lorlatinib

    • At week 2, week 4, and week 8

    • Periodically after week 8

    Why: Detecting lipid increases early allow for early intervention and decreases risk for other complications.

black man with apple, heart, and weight.
  • Lifestyle modification can help to reduce increases in blood lipids:

    • Reduce dietary fat consumption such as fatty meat or snacks that have trans fats on the label.

    • start light exercise including walking, yoga, and swimming.

    • Manage stress when possible: get enough sleep, ask for help when possible, try meditation.

    Why: lipid management reduces baseline risk and may reduce the degree of drug related lipid increase.

heart with plus sign
  • This is particularly important for patients with a history of cardiovascular disease.

    A cardiovascular consultation can help by:

    • Establishing a goal for ideal cholesterol levels.

    • Checking heart rate, blood pressure, and ECG at baseline.

      • Heart rate should be checked at follow up appointments.

    Why: high cholesterol or triglyceride levels can have an impact on heart function so a cardiologist can help monitor lipid levels and heart function.

Management Strategies

lipid lowering medication pill bottle
  • Lipid lowering medication should be taken if blood lipid levels are mild or severe:

    Blood lipid levels are mild if:

    • Cholesterol is between 200-300mg/ dL

    • Triglyceride is between 150-300mg/ dL

    Blood lipids are severe if:

    • Cholesterol is between 401-500mg/ dL

    • Triglyceride is between 501-1000 mg/ dL

    * Optimal blood lipid levels are:

    • Cholesterol less than 200mg/ dL

    • Triglycerides less than 150mg/ dL

doctor holding a pause button
  • If severity reaches grade 4, your healthcare team will pause ALKi’s until lipid levels recover to moderate or mild severity:

    • Grade 4 hypercholesterolemia: Cholesterol over 500mg/ dL.

    • Grade 4 hypertriglyceridemia: triglyceride over 1000mg/ dL.

    You may also have to increase or change to a new lipid lowering therapy.

doctor holding an arrow down
  • If severe hypercholesterolemia or hypertriglyceridemia recurs despite maximal lipid-lowering therapy, your healthcare team will reduce 1 dose level of ALKi.

Emergent Symptoms

If you are unsure, it is always safer to seek medical care.
Tell emergency staff you are on an ALK inhibitor for lung cancer.

phone

Call a Healthcare Provider

Call 811 for health advice from a registered nurse OR call your care team

  • New or worsening abdominal discomfort

  • Ongoing nausea or loss of appetite

  • Unusual fatigue

  • Yellowing of the skin or eyes

  • Changes in blood test results (if told by your care team)

ambulance

Visit an Emergency Room

Call 911 or drive to your closest emergency room

Possible heart attack

  • Chest pressure, pain, or heaviness

  • Pain spreading to the neck, jaw, shoulder, arm, or back

  • Sweating

  • Nausea

  • Lightheadedness or fainting

  • Shortness of breath

Possible stroke (F.A.S.T.)

  • F: face drooping

  • A: arm weakness or numbness

  • S: slurred or hard-to-understand speech

  • T: time- act fast and call 911

Possible pancreatitis

  • Severe stomach or upper abdominal pain (may spread to the back)

  • Nausea and vomiting

  • Fever

  • Fast heartbeat

  • Fast or shallow breathing

These symptoms can happen when triglycerides become very high.

Download Hyperlipidemia Info Sheet
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